Cannabinoid Receptor I (CNR1) (NM_016083) Human Tagged ORF Clone
CAT#: RC210397
- TrueORF®
CNR1 (Myc-DDK-tagged)-Human cannabinoid receptor 1 (brain) (CNR1), transcript variant 1
ORF Plasmid: tGFP
"NM_016083" in other vectors (4)
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CNY 5,488.00
Cited in 8 publications. |
CNY 300.00
Specifications
Product Data | |
Type | Human Tagged ORF Clone |
Tag | Myc-DDK |
Synonyms | CANN6; CB-R; CB1; CB1A; CB1K5; CB1R; CNR |
Vector | pCMV6-Entry |
E. coli Selection | Kanamycin (25 ug/mL) |
Mammalian Cell Selection | Neomycin |
Sequence Data |
>RC210397 representing NM_016083
Red=Cloning site Blue=ORF Green=Tags(s) TTTTGTAATACGACTCACTATAGGGCGGCCGGGAATTCGTCGACTGGATCCGGTACCGAGGAGATCTGCC GCCGCGATCGCC ATGAAGTCGATCCTAGATGGCCTTGCAGATACCACCTTCCGCACCATCACCACTGACCTCCTGTACGTGG GCTCAAATGACATTCAGTACGAAGACATCAAAGGTGACATGGCATCCAAATTAGGGTACTTCCCACAGAA ATTCCCTTTAACTTCCTTTAGGGGAAGTCCCTTCCAAGAGAAGATGACTGCGGGAGACAACCCCCAGCTA GTCCCAGCAGACCAGGTGAACATTACAGAATTTTACAACAAGTCTCTCTCGTCCTTCAAGGAGAATGAGG AGAACATCCAGTGTGGGGAGAACTTCATGGACATAGAGTGTTTCATGGTCCTGAACCCCAGCCAGCAGCT GGCCATTGCAGTCCTGTCCCTCACGCTGGGCACCTTCACGGTCCTGGAGAACCTCCTGGTGCTGTGCGTC ATCCTCCACTCCCGCAGCCTCCGCTGCAGGCCTTCCTACCACTTCATCGGCAGCCTGGCGGTGGCAGACC TCCTGGGGAGTGTCATTTTTGTCTACAGCTTCATTGACTTCCACGTGTTCCACCGCAAAGATAGCCGCAA CGTGTTTCTGTTCAAACTGGGTGGGGTCACGGCCTCCTTCACTGCCTCCGTGGGCAGCCTGTTCCTCACA GCCATCGACAGGTACATATCCATTCACAGGCCCCTGGCCTATAAGAGGATTGTCACCAGGCCCAAGGCCG TGGTGGCGTTTTGCCTGATGTGGACCATAGCCATTGTGATCGCCGTGCTGCCTCTCCTGGGCTGGAACTG CGAGAAACTGCAATCTGTTTGCTCAGACATTTTCCCACACATTGATGAAACCTACCTGATGTTCTGGATC GGGGTCACCAGCGTACTGCTTCTGTTCATCGTGTATGCGTACATGTATATTCTCTGGAAGGCTCACAGCC ACGCCGTCCGCATGATTCAGCGTGGCACCCAGAAGAGCATCATCATCCACACGTCTGAGGATGGGAAGGT ACAGGTGACCCGGCCAGACCAAGCCCGCATGGACATTAGGTTAGCCAAGACCCTGGTCCTGATCCTGGTG GTGTTGATCATCTGCTGGGGCCCTCTGCTTGCAATCATGGTGTATGATGTCTTTGGGAAGATGAACAAGC TCATTAAGACGGTGTTTGCATTCTGCAGTATGCTCTGCCTGCTGAACTCCACCGTGAACCCCATCATCTA TGCTCTGAGGAGTAAGGACCTGCGACACGCTTTCCGGAGCATGTTTCCCTCTTGTGAAGGCACTGCGCAG CCTCTGGATAACAGCATGGGGGACTCGGACTGCCTGCACAAACACGCAAACAATGCAGCCAGTGTTCACA GGGCCGCAGAAAGCTGCATCAAGAGCACGGTCAAGATTGCCAAGGTAACCATGTCTGTGTCCACAGACAC GTCTGCCGAGGCTCTG ACGCGTACGCGGCCGCTCGAGCAGAAACTCATCTCAGAAGAGGATCTGGCAGCAAATGATATCCTGGATT ACAAGGATGACGACGATAAGGTTTAA >RC210397 representing NM_016083
Red=Cloning site Green=Tags(s) MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQEKMTAGDNPQL VPADQVNITEFYNKSLSSFKENEENIQCGENFMDIECFMVLNPSQQLAIAVLSLTLGTFTVLENLLVLCV ILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFIDFHVFHRKDSRNVFLFKLGGVTASFTASVGSLFLT AIDRYISIHRPLAYKRIVTRPKAVVAFCLMWTIAIVIAVLPLLGWNCEKLQSVCSDIFPHIDETYLMFWI GVTSVLLLFIVYAYMYILWKAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILV VLIICWGPLLAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQ PLDNSMGDSDCLHKHANNAASVHRAAESCIKSTVKIAKVTMSVSTDTSAEAL TRTRPLEQKLISEEDLAANDILDYKDDDDKV |
Restriction Sites | SgfI-MluI Cloning Scheme for this gene Plasmid Map |
ACCN | NM_016083 |
ORF Size | 1416 bp |
OTI Disclaimer | The molecular sequence of this clone aligns with the gene accession number as a point of reference only. However, individual transcript sequences of the same gene can differ through naturally occurring variations (e.g. polymorphisms), each with its own valid existence. This clone is substantially in agreement with the reference, but a complete review of all prevailing variants is recommended prior to use. More info |
OTI Annotation | This clone was engineered to express the complete ORF with an expression tag. Expression varies depending on the nature of the gene. |
Product Components | The ORF clone is ion-exchange column purified and shipped in a 2D barcoded Matrix tube containing 10ug of transfection-ready, dried plasmid DNA (reconstitute with 100 ul of water). |
Reconstitution | 1. Centrifuge at 5,000xg for 5min. 2. Carefully open the tube and add 100ul of sterile water to dissolve the DNA. 3. Close the tube and incubate for 10 minutes at room temperature. 4. Briefly vortex the tube and then do a quick spin (less than 5000xg) to concentrate the liquid at the bottom. 5. Store the suspended plasmid at -20°C. The DNA is stable for at least one year from date of shipping when stored at -20°C. |
Reference Data | |
RefSeq | NM_016083.6 |
RefSeq Size | 5486 bp |
RefSeq ORF | 1419 bp |
Locus ID | 1268 |
UniProt ID | P21554 |
Domains | 7tm_1 |
Protein Families | Druggable Genome, GPCR, Transmembrane |
Protein Pathways | Neuroactive ligand-receptor interaction |
MW | 52.7 kDa |
Gene Summary | This gene encodes one of two cannabinoid receptors. The cannabinoids, principally delta-9-tetrahydrocannabinol and synthetic analogs, are psychoactive ingredients of marijuana. The cannabinoid receptors are members of the guanine-nucleotide-binding protein (G-protein) coupled receptor family, which inhibit adenylate cyclase activity in a dose-dependent, stereoselective and pertussis toxin-sensitive manner. The two receptors have been found to be involved in the cannabinoid-induced CNS effects (including alterations in mood and cognition) experienced by users of marijuana. Multiple transcript variants encoding two different protein isoforms have been described for this gene. [provided by RefSeq, May 2009] |
Citations (8)
The use of this cDNA Clones has been cited in the following citations: |
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Rotenoids and Other Specialized Metabolites from the Roots of Mirabilis multiflora: Opioid and Cannabinoid Receptor Radioligand Binding Affinities
,Sharma, VK;Srivedavyasasri, R;Ali, Z;Zjawiony, JK;Ross, SA;Ferreira, D;Ashpole, N;Khan, IA;,
Journal of natural products
,PubMed ID 33734684
[CNR1]
|
Structure-Based Identification of Potent Natural Product Chemotypes as Cannabinoid Receptor 1 Inverse Agonists
,Pandey, P;Roy, KK;Liu, H;Ma, G;Pettaway, S;Alsharif, WF;Gadepalli, RS;Rimoldi, JM;McCurdy, CR;Cutler, SJ;Doerksen, RJ;,
Molecules
,PubMed ID 30322136
[CNR1]
|
Secondary metabolites isolated fromPinus roxburghiiand interpretation of their cannabinoid and opioid binding properties by virtual screening andin vitrostudies
,Labib, RM;Srivedavyasasri, R;Youssef, FS;Ross, SA;,
Saudi Pharm J
,PubMed ID 29556136
[CNR1]
|
Development of a Δ9-Tetrahydrocannabinol Amino Acid-Dicarboxylate Prodrug With Improved Ocular Bioavailability
,Adelli, GR;Bhagav, P;Taskar, P;Hingorani, T;Pettaway, S;Gul, W;ElSohly, MA;Repka, MA;Majumdar, S;,
Invest. Ophthalmol. Vis. Sci.
,PubMed ID 28399267
[CNR1]
|
Pharmacological characterization of emerging synthetic cannabinoids in HEK293T cells and hippocampal neurons.
,null,
European journal of pharmacology
,PubMed ID 27260125
[CNR1]
|
Selective Cannabinoid Receptor-1 Agonists Regulate Mast Cell Activation in an Oxazolone-Induced Atopic Dermatitis Model
,null,
Annals of Dermatology
,PubMed ID 26848215
[CNR1]
|
Topical cannabinoid receptor 1 agonist attenuates the cutaneous inflammatory responses in oxazolone-induced atopic dermatitis model
,Kim, HJ;Kim, B;Park, BM;Jeon, JE;Lee, SH;Mann, S;Ahn, SK;Hong, SP;Jeong, SK;,
Int. J. Dermatol.
,PubMed ID 26095080
[CNR1]
|
Flavonoids from Perovskia atriplicifolia and Their in Vitro Displacement of the Respective Radioligands for Human Opioid and Cannabinoid Receptors
,Tarawneh, A;León, F;Pettaway, S;Elokely, KM;Klein, ML;Lambert, J;Mansoor, A;Cutler, SJ;,
J. Nat. Prod.
,PubMed ID 26035635
[CNR1]
|
Documents
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Resources
Other Versions
SKU | Description | Size | Price |
---|---|---|---|
RC210397L3 | Lenti-ORF clone of CNR1 (Myc-DDK-tagged)-Human cannabinoid receptor 1 (brain) (CNR1), transcript variant 1 |
CNY 7,888.00 |
|
RC210397L4 | Lenti-ORF clone of CNR1 (mGFP-tagged)-Human cannabinoid receptor 1 (brain) (CNR1), transcript variant 1 |
CNY 7,888.00 |
|
RG210397 | CNR1 (tGFP-tagged) - Human cannabinoid receptor 1 (brain) (CNR1), transcript variant 1 |
CNY 7,088.00 |
|
SC111611 | CNR1 (untagged)-Human cannabinoid receptor 1 (brain) (CNR1), transcript variant 1 |
CNY 5,488.00 |
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